| CAT # | Magaca Alaabta | Sharaxaada |
| CPD100616 | Emricasan | Emricasan, oo sidoo kale loo yaqaan IDN 6556 iyo PF 03491390, waa kaspase-ka-hortagga fasalka koowaad ee tijaabooyinka bukaan-socodka ee daaweynta cudurrada beerka. Emricasan (IDN-6556) waxay hoos u dhigtaa dhaawaca beerka iyo fibrosis ee qaabka murka ee steatohepatitis-ka aan khamriga ahayn. IDN6556 waxay sahlaysa ku-oolaynta gasiiradda yar ee gasiirada porcine islet model autotransplant. IDN-6556 afka laga yaabaa inay hoos u dhigto hawlaha aminotransferase ee bukaanada qaba cagaarshow C dabadheeraad ah. PF-03491390 afka laga maamulo ayaa lagu hayaa beerka muddo dheer oo leh soo-gaadhis nidaamsan oo hooseeya, taasoo saameyn ku leh hepatoprotective oo ka dhan ah dhaawaca beerka ee alfa-fas-ku keeno qaabka jiirka . |
| CPD100615 | Q-VD-Oph | QVD-OPH, oo sidoo kale loo yaqaan Quinoline-Val-Asp-Difluorophenoxymethylketone, waa spectrum caspase inhibitor ballaaran oo leh sifooyin antiapoptotic awood leh. Q-VD-OPh waxay ka hortagtaa istaroogga dhallaanka ee jiirka P7: doorka jinsiga. Q-VD-OPh waxay leedahay saameyn liddi ku ah leukemia-ga waxayna la falgeli kartaa fiitamiin D-ga analogga ah si loo kordhiyo calaamadaha HPK1 ee unugyada AML. Q-VD-OPh waxay hoos u dhigtaa apoptosis-ka dhaawaca ah waxayna wanaajisaa soo kabashada shaqada dhabarka ee jiirka ka dib dhaawaca laf dhabarta |
| CPD100614 | Z-DEVD-FMK | Z-DEVD-fmk waa unug-meel-marin karo, horjooge aan laga noqon karin ee caspase-3. Caspase-3 waa cysteinyl aspartate-gaar ah protease kaas oo ka ciyaara doorka dhexe ee apoptosis. |
| CPD100613 | Z-IETD-FMK | MDK4982, oo sidoo kale loo yaqaan Z-IETD-FMK, waa awood xoog leh, unug-wareejin, horjooge aan la bedeli karin ee kaspase-8 iyo granzyme B., Caspase-8 Inhibitor II waxay xakameysaa dhaqdhaqaaqa noolaha ee Caspase-8. MDK4982 waxay si wax ku ool ah u joojisaa fayraska hargabka apoptosis ee unugyada HeLa. MDK4982 sidoo kale waxay joojisaa granzyme B. MDK4982 waxay leedahay CAS # 210344-98-2. |
| CPD100612 | Z-VAD-FMK | Z-VAD-FMK waa unug-meel-marin karo, xannibaadaha pan-caspase aan laga noqon karin. Z-VAD-FMK waxay joojisaa habaynta kasbaska iyo soo-saarka apoptosis ee unugyada burooyinka ee vitro (IC50 = 0.0015 - 5.8 mM). |
| CPD100611 | Belnacasan | Belnacasan, oo sidoo kale loo yaqaan VX-765, waxaa loogu talagalay in lagu xakameeyo Caspase, taas oo ah enzyme xakameynaya jiilka laba cytokines, IL-1b iyo IL-18. VX-765 ayaa la tusay inay joojiso suuxdinta degdega ah ee moodooyinka hore. Intaa waxaa dheer, VX-765 waxay muujisay firfircoonida moodooyinka hore ee suuxdinta dabadheeraad ah. VX-765 ayaa lagu qiyaasey in ka badan 100 bukaan oo ku jira marxaladda-I iyo marxaladda-IIa tijaabooyinka bukaan-socodka ee la xiriira cudurrada kale, oo ay ku jiraan 28-maalmood-IIa tijaabo caafimaad ee bukaannada qaba cudurka psoriasis. Waxay dhammaysay wejigii daawaynta ee wajiga-IIa tijaabada caafimaad ee VX-765 taas oo diiwaangelisay ku dhawaad 75 bukaan oo qaba suuxdin u adkaysta. Laba-indho-indho la'aan, randomized, tijaabada bukaan-socod-koontarool ee placebo waxaa loogu talagalay in lagu qiimeeyo badbaadada, dulqaadka iyo dhaqdhaqaaqa bukaan-socodka ee VX-765. |
