I-GLP-1R

IKATI # Igama Lomkhiqizo Incazelo
I-CPD100594 TT15 I-TT15 iyi-agonist ye-GLP-1R.
I-CPD100593 VU0453379 I-VU0453379 iyi-CNS-penetrant glucagon-like peptide 1 receptor (GLP-1R) positive allosteric module (PAM)
I-CPD100592 PF-06882961 I-PF-06882961 iyi-agonist enamandla, ngomlomo ye-bioavailable ye-glucagon-like peptide-1 receptor (GLP-1R).
I-CPD100591 PF-06372222 I-PF-06372222 iyi-molecule encane ene-negative allosteric modulator (NAM) ye-glucagon receptor (GCGR). Ama-Antagonists e-GCGR angase abe usizo ekwelapheni uhlobo 2 lwesifo sikashukela ngoba alawula amazinga kashukela ku-plasma ngokunciphisa noma ngokunciphisa ukukhiqizwa kwe-glucose esibindini ngokusayina esibindini, emisipha ebushelelezi yamathumbu, izinso, ubuchopho, nezicubu ze-adipose. I-PF-06372222 iphinde ibe ngumphikisi we-glucagon-like peptide-1 receptor GLP-1R, evimbela ukukhiqizwa kwe-glucagon kanye nokukhiqizwa kwe-insulin encike ku-glucose futhi ingase ibe nendima ekukhululweni kwamahomoni okuholela ekucindezelekeni okukhulu nokungapheli kanye nokukhathazeka. Ngokuguqula kabi i-GLP-1R, i-PF-06372222 ingaphatha uhlobo 2 lwesifo sikashukela kanye nengcindezi nokukhathazeka.
I-CPD100590 I-NNC0640 I-NNC0640 iyimoduli ye-allosteric engalungile ye-glucagon-like peptide-1 receptor (GLP-1R).
I-CPD100589 I-HTL26119 I-HTL26119 iyinoveli ephikisana ne-allosteric ye-glucagon-like peptide-1 receptor (GLP-1R).
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