| CAT # | Sunan samfur | Bayani |
| Saukewa: CPD100594 | TT15 | TT15 agonist ne na GLP-1R. |
| Saukewa: CPD100593 | Farashin 0453379 | VU0453379 shine CNS-mai shiga glucagon-kamar peptide 1 mai karɓa (GLP-1R) tabbataccen allosteric modulator (PAM) |
| Saukewa: CPD100592 | Saukewa: PF-06882961 | PF-06882961 mai ƙarfi ne mai ƙarfi, mai haɓakawa na baka na mai karɓar glucagon-kamar peptide-1 (GLP-1R). |
| Saukewa: CPD100591 | Saukewa: PF-0637222 | PF-06372222 ƙananan ƙwayoyin cuta mara kyau na allosteric modulator (NAM) na mai karɓar glucagon (GCGR). Masu adawa da GCGR na iya taimakawa wajen magance nau'in ciwon sukari na 2 saboda suna daidaita matakan glucose na plasma ta hanyar raguwa ko rage yawan samar da glucose na hanta ta hanyar sigina a cikin hanta, tsoka mai santsi na hanji, koda, kwakwalwa, da adipose tissue. PF-06372222 kuma mai adawa ne ga mai karɓar glucagon-kamar peptide-1 GLP-1R, wanda ke hana ƙwayar glucagon da siginar insulin-dogara kuma yana iya taka rawa a cikin sakin hormonal wanda ke haifar da matsananciyar damuwa da damuwa. Ta hanyar canza GLP-1R mara kyau, PF-06372222 na iya magance nau'in ciwon sukari na 2 da damuwa da damuwa. |
| Saukewa: CPD100590 | NNC0640 | NNC0640 shine mummunan allosteric modulator na glucagon-kamar peptide-1 mai karɓa (GLP-1R). |
| Saukewa: CPD100589 | Saukewa: HTL26119 | HTL26119 sabon allosteric antagonist na mai karɓar glucagon-kamar peptide-1 (GLP-1R). |
