| KATSE # | Lebitso la Sehlahiswa | Tlhaloso |
| CPD100594 | TT15 | TT15 ke agonist ea sehlopha sa GLP-1R. |
| CPD100593 | VU0453379 | VU0453379 ke CNS-penetrant glucagon-like peptide 1 receptor (GLP-1R) positive allosteric modulator (PAM) |
| CPD100592 | PF-06882961 | PF-06882961 ke agonist e matla, ea molomo ea bioavailable ea glucagon-like peptide-1 receptor (GLP-1R). |
| CPD100591 | PF-06372222 | PF-06372222 ke molek'hule e nyane ea allosteric modulator (NAM) ea glucagon receptor (GCGR). Bahanyetsi ba GCGR ba ka thusa ho alafa lefu la tsoekere la mofuta oa 2 hobane ba laola maemo a tsoekere ea plasma ka ho fokotsa kapa ho liehisa tlhahiso ea tsoekere ea sebete ka ho hlahisa sebete, mesifa e boreleli ea mala, liphio, boko le lisele tsa adipose. PF-06372222 hape ke mohanyetsi oa glucagon-like peptide-1 receptor GLP-1R, e thibelang secretion ea glucagon le secretion ea insulin e itšetlehileng ka tsoekere 'me e ka boela ea bapala karolo ea ho lokolloa ha li-hormone ho lebisang khatellong e matla le e sa foleng le matšoenyeho. Ka ho fetola GLP-1R hampe, PF-06372222 e ka phekola lefu la tsoekere la mofuta oa 2 le khatello ea maikutlo le matšoenyeho. |
| CPD100590 | NNC0640 | NNC0640 ke modulator e mpe ea allosteric ea glucagon-like peptide-1 receptor (GLP-1R). |
| CPD100589 | HTL26119 | HTL26119 ke mohanyetsi oa "allosteric" oa "glucagon-like peptide-1 receptor" (GLP-1R). |
