| MPAKA # | Dzina lazogulitsa | Kufotokozera |
| CPD100594 | TT15 | TT15 ndi agonist wa GLP-1R. |
| CPD100593 | VU0453379 | VU0453379 ndi CNS-lolowera glucagon-ngati peptide 1 receptor (GLP-1R) positive allosteric modulator (PAM) |
| CPD100592 | PF-06882961 | PF-06882961 ndi agonist wamphamvu, wopezeka pakamwa wa glucagon-ngati peptide-1 receptor (GLP-1R). |
| CPD100591 | PF-06372222 | PF-06372222 ndi yaing'ono-molecule negative allosteric modulator (NAM) ya glucagon receptor (GCGR). Otsutsa a GCGR atha kukhala othandiza pochiza matenda a shuga a mtundu wa 2 chifukwa amawongolera kuchuluka kwa shuga m'magazi mwa kuchepetsa kapena kuchedwetsa kupanga kwa shuga m'chiwindi mwa kuwonetsa chiwindi, minofu yosalala ya m'matumbo, impso, ubongo, ndi minofu ya adipose. PF-06372222 imalimbananso ndi glucagon-ngati peptide-1 receptor GLP-1R, yomwe imalepheretsa katulutsidwe ka glucagon komanso kutulutsa kwa insulin yodalira shuga ndipo imathanso kutenga nawo gawo pakutulutsa kwa mahomoni kumabweretsa kupsinjika kwakukulu komanso kosatha komanso nkhawa. Posintha molakwika GLP-1R, PF-06372222 imatha kuchiza matenda amtundu wa 2 komanso kupsinjika ndi nkhawa. |
| CPD100590 | NNC0640 | NNC0640 ndi allosteric modulator yoyipa ya glucagon-ngati peptide-1 receptor (GLP-1R). |
| CPD100589 | HTL26119 | HTL26119 ndi buku la allosteric antagonist wa glucagon-ngati peptide-1 receptor (GLP-1R). |
