GLP-1R

CAT # Magaca Alaabta Sharaxaada
CPD100594 TT15 TT15 waa agonist ee GLP-1R.
CPD100593 VU0453379 VU0453379 waa CNS-guulaysata glucagon-sida peptide 1 reseptor (GLP-1R) modulator togan (PAM)
CPD100592 PF-06882961 PF-06882961 waa agonist xoog leh oo afka laga heli karo oo ah glucagon-like peptide-1 reseptor (GLP-1R).
CPD100591 PF-06372222 PF-06372222 waa unug yar-molecule negative allosteric modulator (NAM) ee glucagon receptor (GCGR). Ka soo horjeeda GCGR waxaa laga yaabaa inay ku caawiso daaweynta nooca 2 ee sonkorowga mellitus sababtoo ah waxay nidaamiyaan heerarka gulukooska balaasmaha iyagoo hoos u dhigaya ama hoos u dhigaya wax soo saarka gulukooska beerka iyagoo calaamadeynaya beerka, muruqa siman ee mindhicirka, kelyaha, maskaxda, iyo unugyada adipose. PF-06372222 sidoo kale waa ka soo horjeeda glucagon-like peptide-1 reseptor GLP-1R, kaas oo joojiya dheecaanka glucagon iyo dheecaanka insulin-ku-tiirsan ee gulukooska waxana laga yaabaa inay door ka ciyaaraan sii-deynta hoormoonka taasoo keenta walaac ba'an oo dabadheeraad ah iyo walaac. Iyada oo si xun u beddeleysa GLP-1R, PF-06372222 waxay daweyn kartaa nooca 2 ee sonkorowga mellitus iyo walbahaarka iyo walaaca.
CPD100590 NNC0640 NNC0640 waa modulator allosteric taban ee glucagon-like peptide-1 reseptor (GLP-1R).
CPD100589 HTL26119 HTL26119 waa iska soo horjeedka cusub ee allosteric antagonist ee glucagon-like peptide-1 reseptor (GLP-1R).
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