GLP-1R

CAT # Ingoa Hua Whakaahuatanga
CPD100594 TT15 Ko te TT15 he agonist o te GLP-1R.
CPD100593 VU0453379 Ko te VU0453379 he kaikawe peptide 1 rite ki te glucagon-penetrant CNS (GLP-1R) (GLP-1R) totika allosteric modulator (PAM)
CPD100592 PF-06882961 Ko te PF-06882961 he agonist kaha, karekau-a-waha o te kaikawe peptide-1 rite ki te glucagon (GLP-1R).
CPD100591 PF-06372222 Ko te PF-06372222 he iti-ngota ngota kino allosteric modulator (NAM) o te kaikawe glucagon (GCGR). Ka awhina pea nga kaiwhaiwhai o te GCGR ki te rongoa i te mate huka momo 2 na te mea ka whakatauhia e ratou nga taumata huka plasma ma te whakaheke, te whakaroa ranei i te hanga huka ate ate ma te tohu i roto i te ate, te uaua maeneene o te whekau, te whatukuhu, te roro, me te kiko adipose. Ko te PF-06372222 ano he kaitukino mo te glucagon-like peptide-1 receptor GLP-1R, e aukati ana i te hunanga o te glucagon me te hunanga o te insulin e whakawhirinaki ana ki te huka, a tera pea ka whai waahi ki te tuku homoni e arai ana i te ahotea me te awangawanga. Ma te whakarereke kino i te GLP-1R, ka taea e PF-06372222 te rongoa mo te mate huka momo 2 me te ahotea me te awangawanga.
CPD100590 NNC0640 Ko te NNC0640 he kaitahuri allosteric kino o te glucagon-rite peptide-1 receptor (GLP-1R).
CPD100589 HTL26119 Ko te HTL26119 he antagonist allosteric hou o te kaikawe peptide-1 rite ki te glucagon (GLP-1R).
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