| Ologbo # | Orukọ ọja | Apejuwe |
| CPD100594 | TT15 | TT15 jẹ agonist ti GLP-1R. |
| CPD100593 | VU0453379 | VU0453379 jẹ CNS-penetrant glucagon-like peptide 1 receptor (GLP-1R) modulator allosteric rere (PAM) |
| CPD100592 | PF-06882961 | PF-06882961 jẹ alagbara, agonist bioavailable ẹnu ti glucagon-like peptide-1 receptor (GLP-1R). |
| CPD100591 | PF-06372222 | PF-06372222 jẹ modulator odi allosteric odi kekere-moleku (NAM) ti olugba glucagon (GCGR). Awọn alatako ti GCGR le ṣe iranlọwọ ni atọju iru 2 diabetes mellitus nitori wọn ṣe ilana awọn ipele glukosi pilasima nipasẹ idinku tabi idinku iṣelọpọ glukosi ẹdọ nipasẹ isamisi ninu ẹdọ, iṣan didan ifun, kidinrin, ọpọlọ, ati àsopọ adipose. PF-06372222 tun jẹ antagonist fun glucagon-like peptide-1 receptor GLP-1R, eyiti o ṣe idiwọ yomijade glucagon ati yomijade insulin ti o gbẹkẹle glukosi ati pe o tun le ṣe ipa ninu itusilẹ homonu ti o yori si aapọn ati aapọn onibaje ati aibalẹ. Nipa iyipada ti ko dara GLP-1R, PF-06372222 le ṣe itọju iru 2 àtọgbẹ mellitus ati aapọn ati aibalẹ. |
| CPD100590 | NNC0640 | NNC0640 jẹ modulator allosteric odi ti olugba glucagon-like peptide-1 (GLP-1R). |
| CPD100589 | HTL26119 | HTL26119 jẹ antagonist allosteric aramada ti olugba glucagon-like peptide-1 (GLP-1R). |
