| CAT # | Khoom npe | Kev piav qhia |
| PIB 100594 | TT15 | TT15 yog agonist ntawm GLP-1R. |
| PIB 100593 | wb 0453379 | VU0453379 yog CNS-penetrant glucagon-zoo li peptide 1 receptor (GLP-1R) zoo allosteric modulator (PAM) |
| PAB 100592 | PF-06882961 | PF-06882961 yog lub zog, qhov ncauj bioavailable agonist ntawm glucagon-zoo li peptide-1 receptor (GLP-1R). |
| PIB 100591 | PF-06372222 | PF-06372222 yog ib qho me me-molecule negative allosteric modulator (NAM) ntawm glucagon receptor (GCGR). antagonists ntawm GCGR yuav pab tau rau kev kho mob hom 2 mob ntshav qab zib mellitus vim tias lawv tswj hwm cov ntshav qabzib hauv cov ntshav los ntawm kev txo qis lossis qeeb cov piam thaj hauv siab los ntawm kev taw qhia hauv daim siab, cov leeg nqaij du, lub raum, hlwb, thiab cov ntaub so ntswg adipose. PF-06372222 kuj yog ib qho antagonist rau glucagon-zoo li peptide-1 receptor GLP-1R, uas inhibits glucagon secretion thiab glucose-dependent insulin secretion thiab kuj tseem tuaj yeem ua lub luag haujlwm hauv hormonal tso tawm ua rau mob hnyav thiab mob ntev thiab ntxhov siab. Los ntawm kev hloov pauv tsis zoo GLP-1R, PF-06372222 tuaj yeem kho hom 2 mob ntshav qab zib mellitus thiab kev ntxhov siab thiab kev ntxhov siab. |
| PIB 100590 | NPO 0640 | NNC0640 yog qhov tsis zoo allosteric modulator ntawm glucagon-zoo li peptide-1 receptor (GLP-1R). |
| PAB 100589 | HTL26119 | HTL26119 yog ib qho tshiab allosteric antagonist ntawm glucagon-zoo li peptide-1 receptor (GLP-1R). |
