I-GLP-1R

CAT # Igama lemveliso Inkcazo
CPD100594 TT15 I-TT15 yi-agonist ye-GLP-1R.
CPD100593 VU0453379 I-VU0453379 yi-CNS-penetrant glucagon-like peptide 1 receptor (GLP-1R) positive allosteric module (PAM)
CPD100592 PF-06882961 I-PF-06882961 inamandla, i-agonist yomlomo ye-bioavailable ye-glucagon-like peptide-1 receptor (GLP-1R).
CPD100591 PF-06372222 PF-06372222 yi-molecule encinci ye-allosteric modulator (NAM) ye-glucagon receptor (GCGR). Abachasi be-GCGR banokuba luncedo ekuphatheni uhlobo lwe-2 yesifo sikashukela ngenxa yokuba balawula amanqanaba e-glucose ye-plasma ngokunciphisa okanye ukunciphisa ukuveliswa kwe-glucose ye-hepatic ngokubonakalisa isibindi, i-intestinal smooth muscle, intso, ingqondo kunye nezicubu ze-adipose. I-PF-06372222 ikwangumchasi we-glucagon-like peptide-1 receptor GLP-1R, enqanda ukukhutshwa kweglucagon kunye ne-glucose exhomekeke kwi-insulin secretion kwaye inokudlala indima ekukhululweni kwehomoni ekhokelela kuxinzelelo olubukhali kunye nolungapheliyo kunye noxinzelelo. Ngokumodareyitha kakubi i-GLP-1R, PF-06372222 inokunyanga uhlobo lwe-2 yesifo sikashukela kunye noxinzelelo kunye noxinzelelo.
CPD100590 NNC0640 I-NNC0640 yimodyuli ye-allosteric engalunganga ye-glucagon-like peptide-1 receptor (GLP-1R).
CPD100589 HTL26119 I-HTL26119 iyiveli ye-allosteric antagonist ye-glucagon-like peptide-1 receptor (GLP-1R).

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