| CAT # | Izina ryibicuruzwa | Ibisobanuro |
| CPD100594 | TT15 | TT15 ni agoniste wa GLP-1R. |
| CPD100593 | VU0453379 | VU0453379 ni glucagon ya CNS-yinjira muri peptide ya peptide 1 yakira (GLP-1R) moderi nziza ya allosteric modulator (PAM) |
| CPD100592 | PF-06882961 | PF-06882961 ni agoniste ikomeye, mu kanwa bioavailable agonist ya glucagon imeze nka peptide-1 yakira (GLP-1R). |
| CPD100591 | PF-06372222 | PF-06372222 ni molekile ntoya ya allosteric modulator (NAM) ya glucagon reseptor (GCGR). Antagonistes ya GCGR irashobora gufasha mukuvura diyabete yo mu bwoko bwa 2 kuko igenga plasma glucose igabanya cyangwa igabanya umuvuduko wa glucose ya hepatike yerekana umwijima, imitsi yoroshye yo munda, impyiko, ubwonko, hamwe na tipusi ya adipose. PF-06372222 nayo irwanya glucagon imeze nka peptide-1 yakira reseptor GLP-1R, ibuza gusohora glucagon hamwe na glucose iterwa na glucose kandi ishobora no kugira uruhare mukurekura imisemburo itera guhangayika bikabije kandi bidakira no guhangayika. Muguhindura nabi GLP-1R, PF-06372222 irashobora kuvura indwara ya diyabete yo mu bwoko bwa 2 hamwe no guhangayika no guhangayika. |
| CPD100590 | NNC0640 | NNC0640 ni moderi mbi ya allosteric modulator ya glucagon imeze nka peptide-1 yakira (GLP-1R). |
| CPD100589 | HTL26119 | HTL26119 nigitabo gishya cya allosteric antagonist ya glucagon imeze nka peptide-1 yakira (GLP-1R). |
