GLP-1R

nwamba # Aha ngwaahịa Nkọwa
CPD100594 TT15 TT15 bụ agonist nke GLP-1R.
CPD100593 VU0453379 VU0453379 bụ CNS-penetrant glucagon-dị ka peptide 1 nnabata (GLP-1R) nti allosteric modulator (PAM)
CPD100592 PF-06882961 PF-06882961 bụ agonist dị ike, nke nwere ike ịpụta glucagon dị ka peptide-1 nnabata (GLP-1R).
CPD100591 PF-06372222 PF-06372222 bụ obere molekul na-adịghị mma allosteric modulator (NAM) nke nnabata glucagon (GCGR). Ndị na-emegide GCGR nwere ike inye aka n'ịgwọ ụdị ọrịa shuga mellitus nke 2 n'ihi na ha na-achịkwa ọkwa glucose plasma site n'ibelata ma ọ bụ na-ebelata mmepụta glucose imeju site n'igosi na imeju, uru ahụ dị nro nke eriri afọ, akụrụ, ụbụrụ, na anụ ahụ adipose. PF-06372222 bụkwa onye na-emegide glucagon-dị ka peptide-1 receptor GLP-1R, nke na-egbochi secretion glucagon na insulin na-adabere na glucose ma nwee ike na-ekere òkè na ntọhapụ homonụ na-eduga na oke nrụgide na nchekasị na-adịghị ala ala. Site n'ịgbanwe GLP-1R na-adịghị mma, PF-06372222 nwere ike ịgwọ ụdị ọrịa shuga mellitus 2 na nchekasị na nchekasị.
CPD100590 NNC0640 NNC0640 bụ ihe na-adịghị mma allosteric modulator nke glucagon-dị ka peptide-1 nnabata (GLP-1R).
CPD100589 HTL26119 HTL26119 bụ onye na-emegide allosteric nke glucagon-dị ka peptide-1 nnabata (GLP-1R).
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