Derazantinib; ARQ-087

Derazantinib; ARQ-087
  • Name: Derazantinib; ARQ-087
  • Catalog No.: CPDB1093
  • CAS No.: 1234356-69-4
  • Molecular Weight: 468.5764
  • Chemical Formula: C29H29FN4O
  • For scientific research only, not for patients.

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    10mg In Stock 800
    100mg In Stock 1200
    500mg In Stock 1800
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    Derazantinib, ARQ-087, ARQ087, ARQ 087, 1234356-69-4

    Solubility: Soluble in DMSO

    Storage: 0 - 4°C for short term (days to weeks), or -20°C for long term (months).


    Derazantinib, also known as ARQ-087, is an orally bioavailable inhibitor of the fibroblast growth factor receptor (FGFR) with potential antineoplastic activity. FGFR inhibitor ARQ 087 binds to and potently inhibits the activity of FGFR subtypes 1, 2 and 3. This may result in the inhibition of FGFR-mediated signal transduction pathways, tumor cell proliferation, tumor angiogenesis and tumor cell death in FGFR-overexpressing tumor cells. FGFR, a receptor tyrosine kinase, is upregulated in many tumor cell types and plays a key role in tumor cellular proliferation, differentiation, angiogenesis and survival.

    Target: FGFR

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