| CAT # | Product Name | Description |
| CPDP800487 | Vopimetostat; TNG-462 | TNG-462 is an orally effective selective PRMT5 inhibitor. |
| 5-bromo-3-(3-methyl-[2,3'-bipyridin]-6′-y... | ||
| CPD109170 | Osavampator; TAK 653; NBI-1065845 | Osavampator (TAK-653) is a novel AMPA receptor positive allosteric modulator. |
| CPDA601746 | Tuspetinib; HM43239 | Tuspinib (HM43239) is a selective FLT3 inhibitor with oral activity. |
| CPDM400101 | (1S,2S)-2-methoxycyclobutan-1-amine hydrochloride | |
| CPDP802494 | LEI 101; LEI 101 hydrochloride; LEI 101 HCl | LEI-101 is an effective, selective, and orally active agonist of the cannabinoid CB2 receptor. |
| CPDS101250 | N-benzyl-2-((2,6-dimethylphenyl)amino)-N,N-diet... | |
| CPD109387 | 2,4(1H,3H)-Pyrimidinedione, 1,5-dimethyl-6-[2-m... | |
| CPD109473 | BB-Cl-Amidine | BB Cl Amidine is an inhibitor of peptidyl arginine deaminase (PAD). |
| CPDP802572 | PHA-408 | PHA 408 (PHA-408) is an effective, selective, and orally active inhibitor of I κ B kinase-2 (IKK-2). |
| CPD109202 | Nirogacestat HBr; Nirogacestat hydrobromide; PF... | Nirogacestat dihydrobromide (PF-3084014 dihydrobromide) It is an effective, orally active, reversible, non competitive, selective gamma secretase inhibitor. |
| CPD109886 | Mesdopetam · 1/2 L-tartrate salt | |
| CPD109325 | Bifluranol | Bifluranol (BX341) has anti androgenic activity. |
| CPD109334 | His121 ARG57; MAGL-IN-4 | MAGL-IN-4 is an orally effective, selective, and reversible inhibitor of monoacylglycerol lipase (MAGL). |
| CPD109174 | TAK041; NBI-1065846; Zelatriazin | Zelatriazin (TAK-041; NBI-1065846) is an effective and selective GPR139 agonist. |
| CPDA601769 | Casdatifanum; Casdatifan; AB521 | Casdaitifan (AB521) is an orally effective HIF-2 α (hypoxia inducible factor 2 α) inhibitor. |
| CPDP801328 | Glecirasib; JAB-21822 | Glecirasib (Compound 1-2; JAB-21822) is an orally active and effective KRAS G12C inhibitor. |
| CPD113014 | BI-4142 | BI-4142 is an effective, highly selective, and orally active HER2 inhibitor. |
| CPD101120 | Ceralasertib; AZD-6738 | Ceralasertib (AZD6738) is an effective ATR kinase inhibitor. |
| CPD100394 | AZD-1390 | AZD1390 is an effective, highly selective, orally bioavailable, and brain permeable ATM inhibitor. |
| CPDA601963 | AZD-8421 | AZD8421 is a selective CDK2 inhibitor with an IC50 of 9 nM. |
| CPDP802413 | AZD-3470 | |
| CPD109435 | Glumetinib; SCC244 | Glumetinib (SCC244) is a highly selective, orally bioavailable, ATP competitive c-Met inhibitor. |
| CPDA602036 | INCB126503 | |
| CPDA601917 | AZD-2389 | AZD2389 is a potent FAP inhibitor with oral activity. |
| CPDA601920 | IAMA6; ARN23746 | IAMA-6 is a selective NKCC1 inhibitor with neuroprotective effects. |
| CPDM400332 | (R)-methyl 2-((S)-2,2-dimethyl-1,3-dioxolan-4-y... | |
| CPD1805 | IACS-010759; IACS-010759 (HCl) | IACS-010759 or IACS-10759 is a potent and selective Oxidative Phosphorylation Inhibitor (IC50 < 10 nM) with potential antineoplastic activity. |
| CPDA600747 | CDK2-IN-73; CDK2-IN-4 | CDK2-IN-73 is a potent and highly selective CDK2 inhibitor. |
| CPD114044 | 1H-Pyrazole-4-carboxylic acid, 3-(methoxymethyl... |